A synthesis of dibucaine labeled with l"C in the heterocyclic ring is described. starting with isatin and acetic anh~dride-2-~"C as shown in Scheme I. Two deutero analogs, dibucaine-d2 and dibucaine-dg, were also synthesized by the reactions shown in Scheme 11. Dibucaine-dg was synthesized by conden
The synthesis of 14C, 3H and 2H labeled 7-ethoxycoumarins
✍ Scribed by John S. Walsh; Holly E. Mertel; Gerald T. Miwa
- Publisher
- John Wiley and Sons
- Year
- 1983
- Tongue
- French
- Weight
- 266 KB
- Volume
- 20
- Category
- Article
- ISSN
- 0022-2135
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