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Synthesis of PNU-243922 labelled with 14C

✍ Scribed by C. Felicini; E. Fontana; D. Giribone; B. M. Nilsson; K. Österlund; A. Paptchikhine

Publisher
John Wiley and Sons
Year
2002
Tongue
French
Weight
90 KB
Volume
46
Category
Article
ISSN
0022-2135

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✦ Synopsis

Abstract

The arylpiperazine PNU‐243922 (1) has been labelled with ^14^C. A two‐step sequence starting from the ^14^C labelled alcohol 6a led to radiochemically pure (>98%) [^14^C]PNU‐243922 with a specific activity of 546 MBq/mmol Copyright © 2002 John Wiley & Sons, Ltd.

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