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Synthesis of PHA-690509 labelled with 14C

✍ Scribed by E. Fontana; D. Giribone; C. Felicini

Publisher: John Wiley and Sons
Year: 2007
Tongue: French
Weight: 84 KB
Volume: 50
Category: Article
ISSN: 0022-2135
DOI: 10.1002/jlcr.1253

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✦ Synopsis

Abstract

PHA‐690509, a cyclin‐dependent kinase A inhibitor, has been labelled with carbon‐14. [^14^C]PHA‐690509 was obtained via a three‐step procedure in 10% overall radiochemical yield starting from [^14^C]thiourea 3. Copyright © 2007 John Wiley & Sons, Ltd.

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