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Synthesis of new perhydro-(1,4)-diazepin-2-ones as constrained peptidomimetics

✍ Scribed by André Nouvet; Frédéric Lamaty; René Lazaro

Book ID
104258855
Publisher
Elsevier Science
Year
1998
Tongue
French
Weight
168 KB
Volume
39
Category
Article
ISSN
0040-4039

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✦ Synopsis

New access to substituted perhydro-(1,4)-diazepin-2-ones has been developed through either a Mitsunobu reaction or an amide bond formation for the eyclisation key step.

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