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Synthesis of encainide-13C hydrochloride from 2-nitrobenzaldehyde-formyl-13C

โœ Scribed by Porter C. Johnson; Robert R. Covington

Publisher
John Wiley and Sons
Year
1982
Tongue
French
Weight
213 KB
Volume
19
Category
Article
ISSN
0022-2135

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โœฆ Synopsis

Abstract

A tacile synthesis of 2โ€nitrobenzaldehydeโ€formylโ€^13^C was developed. This compound was converted to the labelled antiarrhythmic agent, encainideโ€^13^C hydrochloride, 4โ€methoxyโ€Nโ€[2โ€[2โ€(1โ€methylโ€2โ€piperidinyl)ethylโ€1โ€^13^C]phenyl]benzamide hydrochloride.

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