✦ LIBER ✦

Synthesis of 14C-bucromarone succinate and hydrochloride

✍ Scribed by Colette Nicolas; Michel Verny; Jean-Claude Maurizis; Marc Payard; Michel Faurie

Publisher: John Wiley and Sons
Year: 1986
Tongue: French
Weight: 287 KB
Volume: 23
Category: Article
ISSN: 0022-2135
DOI: 10.1002/jlcr.2580230806

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✦ Synopsis

[2]

[3]

[4]N dibutylamino propoxy)

3,S-dirnethyl benzoyl] chromone, was synthesized from (U-14C) oxalic acid. The labelling takes place at the first step of the synthesis, and allowed the obtention o f -14C-Bucromarone succinate, with a specific activity o f 7.45 mCi/mmol, i.e. 275.6 MBq/mmol ; -14C-Bucromarone hydrochloride, with a specific activity o f 7.5 mCi/mmol, i.e. 277.5 MBq/mmol.

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