## Abstract Condensation of phenylazo‐β‐ketoamide **4** with oxymorphone **5** afforded an __m__‐iodophenylpyrrolomorphinan (__m__‐IPPM) **6** mediated by elemental zinc in acetic acid/sodium acetate buffer. __m__‐IPPM **6** is a novel opioid receptor agonist (__K__~i~ = 4.53 nM for DOP) with high
Synthesis and in vivo PET imaging studies with [11C]BU4033, a potential delta opioid imaging agent
✍ Scribed by Michael R. Kilbourn; D. Donnelly; S.M. Husbands; B. Greedy; J.H. Woods; J.R. Traynor
- Book ID
- 118491190
- Publisher
- Elsevier Science
- Year
- 2008
- Tongue
- English
- Weight
- 57 KB
- Volume
- 41
- Category
- Article
- ISSN
- 1053-8119
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