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Reparation of 3H-, and 14C-labeled ethylmorphine

✍ Scribed by Yul Yost; Jordan L. Holtzman

Publisher: John Wiley and Sons
Year: 1981
Tongue: French
Weight: 179 KB
Volume: 18
Category: Article
ISSN: 0022-2135
DOI: 10.1002/jlcr.2580181212

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✦ Synopsis

Abstract

7,8‐Didehydro‐4,5‐epoxy‐3‐ethoxy‐17‐methyl(^3^H)‐, and −17‐methyl (^14^C)morphinan‐6‐ol were prepared by substituting the N‐methyl group with/^a^carbphenoxy group which was then either reduced with LiAl^3^H~4~ or removed to remethylate the N‐atom with ^14^CH~3~I.

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