The preparation of the 61-specific ligand 7-benzylidenenaltrexone (BNTX), labeled with tritium at high specific activity (14.4 Ciimmol) was prepared in 33% yield and >98% purity by the aldol condensation of high specific activity [15,1 6-3H]naltrexone with benzaldehyde at high dilution.
Preparation of iodo derivatives and high specific activity 3H synthetic human gastrin I
✍ Scribed by Girma, J.P.; Morgat, J.L.; Fromageot, P.; Dubrasquet, M.; Accary, J.P.; Vatier, J.; Bonfils, S.
- Book ID
- 121918032
- Publisher
- Elsevier Science
- Year
- 1974
- Tongue
- English
- Weight
- 383 KB
- Volume
- 56
- Category
- Article
- ISSN
- 0300-9084
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