The preparation of the 61-specific ligand 7-benzylidenenaltrexone (BNTX), labeled with tritium at high specific activity (14.4 Ciimmol) was prepared in 33% yield and >98% purity by the aldol condensation of high specific activity [15,1 6-3H]naltrexone with benzaldehyde at high dilution.
Preparation OF [7, 8, 19, 20 - 3H] Naloxone of high specific activity
✍ Scribed by G. Toth; M. Kramer; F. Sirokman; A. Borsodi; A. Ronai
- Publisher
- John Wiley and Sons
- Year
- 1982
- Tongue
- French
- Weight
- 321 KB
- Volume
- 19
- Category
- Article
- ISSN
- 0022-2135
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