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Pharmacological characterization of a novel phosphodiesterase type 5 (PDE5) inhibitor lodenafil carbonate on human and rabbit corpus cavernosum

โœ Scribed by Haroldo A. Toque; Cleber E. Teixeira; Raquel Lorenzetti; Cristina E. Okuyama; Edson Antunes; Gilberto De Nucci


Book ID
113587725
Publisher
Elsevier Science
Year
2008
Tongue
English
Weight
713 KB
Volume
591
Category
Article
ISSN
0014-2999

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Pharmacological characterization of the
โœ Gilberto De Nucci; Raquel Lorenzetti; Cristina E Okuyama; Juliana S Baracat; Jos ๐Ÿ“‚ Article ๐Ÿ“… 2007 ๐Ÿ› BioMed Central ๐ŸŒ English โš– 785 KB

## Background Nitrergic nerves and endothelial cells release nitric oxide (NO) in the corpus cavernosum (CC), a key mediator that stimulates soluble guanylyl cyclase to increase cGMP levels and cause penile erection. Phosphodiesterase 5 (PDE5) inhibitors, such as sildenafil, prolong NO effects by