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Labelling of 1-benzyl-1- (3′ -dimethylaminopropoxy)- cycloheptane, fumarate with tritium

✍ Scribed by D. Banfi; G. Zolyomi; L. Pallos

Publisher
John Wiley and Sons
Year
1973
Tongue
French
Weight
344 KB
Volume
9
Category
Article
ISSN
0022-2135

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✦ Synopsis

Abstract

In order to complete our previous publications on pharmacokinetics, action mechanism and metabolism studies, the following new, tritium‐labelled derivatives of Halidor have been prepared: 1‐benzyl ‐1‐(3′‐dimethylaminopropoxy) ‐3, 4, 5, 6‐^3^H‐cycloheptane fumarate, 1‐benzyl‐1‐(2′‐^3^H‐3′‐dimethylaminopropoxy)‐cycloheptane fumarate, and 1‐(benzyl‐4‐^3^H)‐(3′‐dimethylaminopropoxy)‐cycloheptane fumarate.

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