## Abstract The α‐hydroxybenzylphosphonates 1a–1j of the antiviral drug 3′‐azido‐2′,3′‐dideoxythymidine 5 (AZT) as potential lipophilic prodrugs were readily accessible in 49% to 87% yield via a four‐step synthetic pathway introducing the modifications in the aromatic ring system in the last step b
✦ LIBER ✦
Homo Dinucleoside-α-hydroxyphosphonate Diesters as Prodrugs of the Antiviral Nucleoside Analogues 2',3'-Dideoxythymidine and 3'-Azido-2',3'-dideoxythymidine
✍ Scribed by Meier, Chris; Habel, Lothar; Laux, Wolfgang; De Clercq, Erik; Balzarini, Jan
- Book ID
- 120466783
- Publisher
- Taylor and Francis Group
- Year
- 1995
- Tongue
- English
- Weight
- 206 KB
- Volume
- 14
- Category
- Article
- ISSN
- 0732-8311
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