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Discovery of (R)-4-(8-Fluoro-2-oxo-1,2-dihydroquinazolin-3(4H)-yl)-N-(3-(7-methyl-1H-indazol-5-yl)-1-oxo-1-(4-(piperidin-1-yl)piperidin-1-yl)propan-2-yl)piperidine-1-carboxamide (BMS-694153): A Potent Antagonist of the Human Calcitonin Gene-Related Peptide Receptor for Migraine with Rapid and Efficient Intranasal Exposure

✍ Scribed by Degnan, Andrew P.; Chaturvedula, Prasad V.; Conway, Charles M.; Cook, Deborah A.; Davis, Carl D.; Denton, Rex; Han, Xiaojun; Macci, Robert; Mathias, Neil R.; Moench, Paul

Book ID: 111651995
Publisher: American Chemical Society
Year: 2008
Tongue: English
Weight: 463 KB
Volume: 51
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm800546t

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