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Design and Synthesis of a Series of (2 R )- N 4 -Hydroxy-2-(3-hydroxybenzyl)- N 1 - [(1 S ,2 R )-2-hydroxy-2,3-dihydro-1 H -inden- 1-yl]butanediamide Derivatives as Potent, Selective, and Orally Bioavailable Aggrecanase Inhibitors †

✍ Scribed by Yao, Wenqing; Wasserman, Zelda R.; Chao, Michael; Reddy, Gade; Shi, Eric; Liu, Rui-Qin; Covington, Maryanne B.; Arner, Elizabeth C.; Pratta, Michael A.; Tortorella, Micky; Magolda, Ronald L.; Newton, Robert; Qian, MingXin; Ribadeneira, Maria D.; Christ, David; Wexler, Ruth R.; Decicco, Carl P.

Book ID: 127233301
Publisher: American Chemical Society
Year: 2001
Tongue: English
Weight: 82 KB
Volume: 44
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm015533c

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