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Design and Pharmacology of N -[(3 R )-1,2,3,4-Tetrahydroisoquinolinium- 3-ylcarbonyl]-(1 R )-1-(4-chlorobenzyl)- 2-[4-cyclohexyl-4-(1 H -1,2,4-triazol- 1-ylmethyl)piperidin-1-yl]-2-oxoethylamine ( 1 ), a Potent, Selective, Melanocortin Subtype-4 Receptor Agonist

✍ Scribed by Sebhat, Iyassu K.; Martin, William J.; Ye, Zhixiong; Barakat, Khaled; Mosley, Ralph T.; Johnston, David B. R.; Bakshi, Raman; Palucki, Brenda; Weinberg, David H.; MacNeil, Tanya; Kalyani, Rubana N.; Tang, Rui; Stearns, Ralph A.; Miller, Randy R.; Tamvakopoulos, Constantin; Strack, Alison M.; McGowan, Erin; Cashen, Doreen E.; Drisko, Jennifer E.; Hom, Gary J.; Howard, Andrew D.; MacIntyre, D. Euan; van der Ploeg, Lex H. T.; Patchett, Arthur A.; Nargund, Ravi P.

Book ID: 121338289
Publisher: American Chemical Society
Year: 2002
Tongue: English
Weight: 132 KB
Volume: 45
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm025539h

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