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Biphenylsulfonamide Endothelin Receptor Antagonists. 4. Discovery of N -[[2‘-[[(4,5-Dimethyl-3-isoxazolyl)amino]sulfonyl]-4-(2-oxazolyl)[1,1‘-biphenyl]- 2-yl]methyl]- N ,3,3-trimethylbutanamide (BMS-207940), A Highly Potent and Orally Active ET A Selective Antagonist

✍ Scribed by Murugesan, Natesan; Gu, Zhengxiang; Spergel, Steven; Young, Marian; Chen, Ping; Mathur, Arvind; Leith, Leslie; Hermsmeier, Mark; Liu, Eddie C.-K.; Zhang, Rongan; Bird, Eileen; Waldron, Tom; Marino, Anthony; Koplowitz, Barry; Humphreys, W. Griffith; Chong, Saeho; Morrison, Richard A.; Webb, Maria L.; Moreland, Suzanne; Trippodo, Nick; Barrish, Joel C.

Book ID: 119995822
Publisher: American Chemical Society
Year: 2003
Tongue: English
Weight: 241 KB
Volume: 46
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm020289q

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