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Biphenylsulfonamide Endothelin Antagonists: Structure−Activity Relationships of a Series of Mono- and Disubstituted Analogues and Pharmacology of the Orally Active Endothelin Antagonist 2‘-Amino- N - (3,4-dimethyl-5-isoxazolyl)-4‘-(2-methylpropyl)[1,1‘-biphenyl]-2-sulfonamide (BMS-187308)

✍ Scribed by Murugesan, Natesan; Gu, Zhengxiang; Stein, Philip D.; Bisaha, Sharon; Spergel, Steve; Girotra, Ravi; Lee, Ving G.; Lloyd, John; Misra, Raj N.; Schmidt, Joan; Mathur, Arvind; Stratton, Leslie; Kelly, Yolanda F.; Bird, Eileen; Waldron, Tom; Liu, Eddie C.-K.; Zhang, Rongan; Lee, Helen; Serafino, Randy; Abboa-Offei, Benoni; Mathers, Parker; Giancarli, Mary; Seymour, Andrea Ann; Webb, Maria L.; Moreland, Suzanne; Barrish, Joel C.; Hunt, John T.

Book ID: 119995826
Publisher: American Chemical Society
Year: 1998
Tongue: English
Weight: 290 KB
Volume: 41
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm970872k

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