✦ LIBER ✦

Unexpected antipsychotic-like activity with the muscarinic receptor ligand (5R,6R)6-(3-propylthio-1,2,5-thiadiazol-4-yl)-1-azabicyclo[3.2.1]octane

✍ Scribed by Frank P Bymaster; Harlan E Shannon; Kurt Rasmussen; Neil W Delapp; Charles H Mitch; John S Ward; David O Calligaro; Thomas S Ludvigsen; Malcolm J Sheardown; Preben H Olesen; Michael D.B Swedberg; Per Sauerberg; Anders Fink-Jensen

Book ID: 114016494
Publisher: Elsevier Science
Year: 1998
Tongue: English
Weight: 405 KB
Volume: 356
Category: Article
ISSN: 0014-2999
DOI: 10.1016/s0014-2999(98)00487-7

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Synthesis of the selective muscarinic ag

Synthesis of the selective muscarinic agonist (3R)-3-(6-chloropyrazin-2-yl)-1-azabicyclo [2.2.2] octane

✍ Ashwood, Michael S.; Gibson, Andrew W.; Houghton, Peter G.; Humphrey, Guy R.; Ro 📂 Article 📅 1995 🏛 Royal Society of Chemistry ⚖ 528 KB

Synthesis and structural determination o

Synthesis and structural determination of stereoisomers of muscarinic ligands of the (3-propylthio-1,2,5-thiadiazol-4-yl)-1-azabicycloalkane type

✍ Preben H. Olesen; Per Sauerberg; Torben G. Petersen; Svend Treppendahl; Bjørn Be 📂 Article 📅 1997 🏛 John Wiley and Sons 🌐 English ⚖ 205 KB 👁 2 views

Methods for the synthesis of each of the four stereoisomers of 6-(3propylthio-1,2,5-thiadiazol-4-yl)-1-azabicyclo[3.2.1]octane (10, 11, 12, and 13) and 3-(3-propylthio-1,2,5-thiadiazol-4-yl)-1-azabicyclo[2.2.1]heptane (18, 19, 20, and 21), and the two stereoisomers of 3-(3-propylthio-1,2,5-thiadiazo

Conformationally Constrained Analogues o

Conformationally Constrained Analogues of the Muscarinic Agonist 3-(4-(Methylthio)-1,2,5-thiadiazol-3-yl)-1,2,5,6-tetrahydro-1-methylpyridine. Synthesis, Receptor Affinity, and Antinociceptive Activity

✍ Sauerberg, Per; Olesen, Preben H.; Sheardown, Malcolm J.; Rimvall, Karin; Thøger 📂 Article 📅 1998 🏛 American Chemical Society 🌐 English ⚖ 193 KB

Antimycotic activity of 6-R-2-(5-nitrofu

Antimycotic activity of 6-R-2-(5-nitrofur-2-yl)-1,3,4,9-tetraazafluorenes

✍ P. A. Pavlov; N. Yu. Basova; P. P. Pavlov 📂 Article 📅 1999 🏛 Springer 🌐 English ⚖ 63 KB

Synthesis of 1-Methyl-5-(pyrazol-3- and

Synthesis of 1-Methyl-5-(pyrazol-3- and -5-yl- and 1,2,4-triazol-3- and 5-yl)-1,2,3,6-tetrahydropyridine Derivatives and Their Evaluation as Muscarinic Receptor Ligands.

✍ Maria Rosaria Del Giudice; Carlo Mustazza; Anna Borioni; Franco Gatta; Khosrow T 📂 Article 📅 2003 🏛 John Wiley and Sons ⚖ 119 KB 👁 1 views

## Abstract For Abstract see ChemInform Abstract in Full Text.

Synthesis of 1-Methyl-5-(pyrazol-3- and

Synthesis of 1-Methyl-5-(pyrazol-3- and -5-yl- and 1, 2, 4-triazol-3- and 5-yl)-1, 2, 3, 6-tetrahydropyridine Derivatives and Their Evaluation as Muscarinic Receptor Ligands

✍ Maria Rosaria Del Giudice; Carlo Mustazza; Anna Borioni; Franco Gatta; Khosrow T 📂 Article 📅 2003 🏛 John Wiley and Sons 🌐 English ⚖ 249 KB 👁 1 views