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Triflates as synthons for the synthesis of lysine analogues

✍ Scribed by Ingo Weber; Pierre Potier; Josiane Thierry

Publisher
Elsevier Science
Year
1999
Tongue
French
Weight
207 KB
Volume
40
Category
Article
ISSN
0040-4039

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✦ Synopsis

A simple synthesis of various 6-amino-2-substitutcd hexanoic acids has been developed starting from lysine via the triflate of 6-amino-2-hydroxy hexanoic acid. The same reactions have also been successfully applied starting from the lysyl-proline sequence. The lysine analogues have been introduced in pseudopeptide sequences by the acylfluoride methodology.

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ChemInform Abstract: Triflates as Syntho
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