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The enantioselective synthesis of LTD4 antagonist L-708,738

✍ Scribed by Daniel R. Sidler; Jess W. Sager; James J. Bergan; Kenneth M. Wells; M. Bhupathy; R.P. Volante

Publisher
Elsevier Science
Year
1997
Tongue
English
Weight
517 KB
Volume
8
Category
Article
ISSN
0957-4166

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✦ Synopsis

An efficient, 9-step synthesis of LTD4 antagonist L-708,738 is described. The asymmetric center is set via a chiral borane reduction.

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