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The Discovery of N -[5-(4-Bromophenyl)-6-[2-[(5-bromo-2-pyrimidinyl)oxy]ethoxy]-4-pyrimidinyl]- N ′-propylsulfamide (Macitentan), an Orally Active, Potent Dual Endothelin Receptor Antagonist

✍ Scribed by Bolli, Martin H.; Boss, Christoph; Binkert, Christoph; Buchmann, Stephan; Bur, Daniel; Hess, Patrick; Iglarz, Marc; Meyer, Solange; Rein, Josiane; Rey, Markus; Treiber, Alexander; Clozel, Martine; Fischli, Walter; Weller, Thomas

Book ID: 118048055
Publisher: American Chemical Society
Year: 2012
Tongue: English
Weight: 607 KB
Volume: 55
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm3009103

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