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Synthesis of a fully protected (2S,3R)-N-(1′,1′-dimethyl-2′- propenyl)-3-hydroxytryptophan from tryptophan

✍ Scribed by Shi-Jun Wen; Hong-Wang Zhang; Zhu-Jun Yao

Publisher
Elsevier Science
Year
2002
Tongue
French
Weight
80 KB
Volume
43
Category
Article
ISSN
0040-4039

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✦ Synopsis

2S,3R)-N-(1%,1%-Dimethyl-2%-propenyl)-3-hydroxytryptophan, a key amino acid of the anti-inflammatory cyclic peptide, cyclomarin C, has been synthesized stereoselectively, with full protection, from L-tryptophan for the first time.

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