## Abstract A simple and convenient laboratory procedure is described by which hordenine (III), labelled at the carbon residing on the benzene ring, can be synthesized by decarboxylation of 3‐ [^14^C]‐tyrosine (1) and subsequent reductive methylation of the resulting tyramine (II).
Synthesis of 4-|2-(dimethylamino) ethyl-2-14C| phenol (hordenine-α-14C)
✍ Scribed by C. A. Russo; E. G. Gros
- Publisher
- John Wiley and Sons
- Year
- 1981
- Tongue
- French
- Weight
- 152 KB
- Volume
- 18
- Category
- Article
- ISSN
- 0022-2135
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✦ Synopsis
Abstract
4‐|2‐(Dimethylamino)ethyl‐2‐^14^C| phenol (hordenine‐α‐^14^C) has been synthesised in three steps from |^14^C|potassium cyanide and p‐benzyloxybenzyl chloride which in turn was obtained in four steps from p‐hydroxybenzoic acid.
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