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Synthesis of 2-deoxy-2-[18F]-fluoro-β-mannosyl [18F]-fluoride as a potential imaging probe for Glycosidases

✍ Scribed by John D. McCarter; Michael J. Adam; Stephen G. Withers


Publisher
John Wiley and Sons
Year
1992
Tongue
French
Weight
221 KB
Volume
31
Category
Article
ISSN
0022-2135

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✦ Synopsis


Abstract

The mechanisms‐based glycosidase inhibitor 2‐deoxy‐2‐[^18^F]‐fluoro‐β‐mannosyl [^18^F]‐fluoride was synthesized and its covalent binding to Agrobacterium β‐glucosidase was demonstrated in vitro.


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