## Abstract Radiolabelled [^14^C]entecavir, (**1**), was prepared in 12 steps from (1S,2R,3S,5R)β3β(benzyloxy)β2β(benzyloxymethyl)β6βoxaβbicyclo[3.1.0]hexane **2**. The chemical yield of [^14^C]entecavir was 14% from the epoxide **2**. Introduction of [^14^C] radiolabel was achieved by elaboration
Synthesis of 14C-radiolabelled tilmicosin
β Scribed by Gary D. Crouse; Norman H. Terando
- Publisher
- John Wiley and Sons
- Year
- 1989
- Tongue
- French
- Weight
- 265 KB
- Volume
- 27
- Category
- Article
- ISSN
- 0022-2135
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