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Synthesis of 14C-labelled 1-methanesulphonyl-3-(1-methyl-5-nitro-1H-imidazol-2-YL)-2-imidazolidinone, (Go 10213)

✍ Scribed by B. Anjaneyulu; R. K. Maller; K. Nagarajan

Publisher
John Wiley and Sons
Year
1983
Tongue
French
Weight
333 KB
Volume
20
Category
Article
ISSN
0022-2135

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✦ Synopsis

E ) , Bombay 400 063, I N D I A F o r pharmacokinetic and metabolism s t u d i e s i n animals and humans, Go 1C213 was l a b e l l e d w i t h carbon-14 a t t h e 2-position o f t h e 5-nitroimidazole r i n g system, i n a n o v e r a l l y i e l d o f 22% s t a r t i n g w i t h potassium[14C]t h i o c y a n a t e . a c t i v i t y o f 4.65 pCi/mg o r 1.34 mCi/mmol.

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