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Synthesis of 14C-labeled inhibitors of monoamine oxidase

✍ Scribed by C. H. Williams

Publisher
John Wiley and Sons
Year
1981
Tongue
French
Weight
190 KB
Volume
18
Category
Article
ISSN
0022-2135

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✦ Synopsis

Abstract

The monoamine oxidase inhibitors pargyline and clorgyline have been synthesized by methylation of the appropriate secondary propargylamines, using [^14^C]dimethyl sulphate. This simple method should be generally applicable to other compounds of this class.

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