A series of analogues of diacylglycerol has been prepared and tested as inhibitors of protein kinase C (PKC). The diketone analogues, 10-hydroxymethyl-8,13-eicosanedione (24), 10-acetoxymethyl-8,13-eicosanedione (25), and 10-methoxymethyl-8,13-eicosanedione (26) each inhibited PKC activated by 2-O-a
โฆ LIBER โฆ
Synthesis and evaluation of iodinated analogs of diacylglycerols as potential probes for protein kinase C
โ Scribed by Strawn, Laurie M.; Martell, Robert E.; Simpson, Robert U.; Leach, Karen L.; Counsell, Raymond E.
- Book ID
- 126434676
- Publisher
- American Chemical Society
- Year
- 1989
- Tongue
- English
- Weight
- 781 KB
- Volume
- 32
- Category
- Article
- ISSN
- 0022-2623
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