✦ LIBER ✦

Synthesis and Characterization of Potent and Selective μ-Opioid Receptor Antagonists, [Dmt 1 , d -2-Nal 4 ]endomorphin-1 (Antanal-1) and [Dmt 1 , d -2-Nal 4 ]endomorphin-2 (Antanal-2)

✍ Scribed by Fichna, Jakub; do-Rego, Jean-Claude; Chung, Nga N.; Lemieux, Carole; Schiller, Peter W.; Poels, Jeroen; Vanden Broeck, Jozef; Costentin, Jean; Janecka, Anna

Book ID: 127201361
Publisher: American Chemical Society
Year: 2007
Tongue: English
Weight: 479 KB
Volume: 50
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm060998u

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

[d-1-Nal4]endomorphin-2 is a potent μ-op

[d-1-Nal4]endomorphin-2 is a potent μ-opioid receptor antagonist in the aequorin luminescence-based calcium assay

✍ Jakub Fichna; Mariola Piestrzeniewicz; Katarzyna Gach; Jeroen Poels; Emmanuel Bu 📂 Article 📅 2006 🏛 Elsevier Science 🌐 English ⚖ 206 KB

Synthesis of benzo[1,2-d;3,4-d′]diimidaz

Synthesis of benzo[1,2-d;3,4-d′]diimidazole and 1H-pyrazolo[4,3-b]pyridine as putative A2A receptor antagonists

✍ Giorgi, Luca; Piersanti, Giovanni; Bartoccini, Francesca; Tarzia, Giorgio; Minet 📂 Article 📅 2007 🏛 Royal Society of Chemistry 🌐 English ⚖ 146 KB

Design and Pharmacology of N -[(3 R )-1,

Design and Pharmacology of N -[(3 R )-1,2,3,4-Tetrahydroisoquinolinium- 3-ylcarbonyl]-(1 R )-1-(4-chlorobenzyl)- 2-[4-cyclohexyl-4-(1 H -1,2,4-triazol- 1-ylmethyl)piperidin-1-yl]-2-oxoethylamine ( 1 ), a Potent, Selective, Melanocortin Subtype-4 Receptor Agonist

✍ Sebhat, Iyassu K.; Martin, William J.; Ye, Zhixiong; Barakat, Khaled; Mosley, Ra 📂 Article 📅 2002 🏛 American Chemical Society 🌐 English ⚖ 132 KB

Design, Synthesis, and SAR of 2-Dialkyla

Design, Synthesis, and SAR of 2-Dialkylamino-4-arylpyrimidines as Potent and Selective Corticotropin-Releasing Factor1 (CRF1) Receptor Antagonists.

✍ Charles Q. Huang; Dimitri E. Grigoriadis; Zhengyu Liu; James R. McCarthy; John R 📂 Article 📅 2004 🏛 John Wiley and Sons ⚖ 62 KB 👁 2 views

1,2,4-Triazol-3-yl-thiopropyl-tetrahydro

1,2,4-Triazol-3-yl-thiopropyl-tetrahydrobenzazepines: A Series of Potent and Selective Dopamine D 3 Receptor Antagonists

✍ Micheli, Fabrizio; Bonanomi, Giorgio; Blaney, Frank E.; Braggio, Simone; Capelli 📂 Article 📅 2007 🏛 American Chemical Society 🌐 English ⚖ 281 KB

Synthesis of Novel Pyrido[3,2- e ][1,2,4

Synthesis of Novel Pyrido[3,2- e ][1,2,4]triazolo[1,5- c ]pyrimidine Derivatives: Potent and Selective Adenosine A 3 Receptor Antagonists

✍ Banda, Veeraswamy; Chandrasekaran, Balakumar; Köse, Meryem; Vielmuth, Christin; 📂 Article 📅 2013 🏛 John Wiley and Sons 🌐 English ⚖ 184 KB