## Abstract Fenobam is a clinically efficacious anxiolytic that acts as metabotropic glutamate receptor 5 (mGlu5) antagonist by binding to an allosteric site. Other mGlu5 receptor antagonists such as MPEP and MTEP bind to the same allosteric site and are efficacious in preclinical models of anxiety
Synthesis and characterization of [3H]-SN56, a novel radioligand for the σ1 receptor
✍ Scribed by James A. Fishback; Christophe Mesangeau; Jacques H. Poupaert; Christopher R. McCurdy; Rae R. Matsumoto
- Book ID
- 113589100
- Publisher
- Elsevier Science
- Year
- 2011
- Tongue
- English
- Weight
- 543 KB
- Volume
- 653
- Category
- Article
- ISSN
- 0014-2999
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