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Synthesis and central nervous system stimulant activity of camphor-1,2,3-triazine fused with diphenylcyclopropenone and camphor-1,2,3-triazine n-oxides

✍ Scribed by Shin-Ichi Nagai; Taisei Ueda

Publisher
Journal of Heterocyclic Chemistry
Year
2000
Tongue
English
Weight
149 KB
Volume
37
Category
Article
ISSN
0022-152X

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✦ Synopsis

Abstract

Reactions of camphor‐1,2,3‐triazine 1 with diphenylcyclopropenone 2 gave two cycloadducts; 6,9‐methanopyrazolo[1,2‐b][1,2,3]benzotriazinones 3–4. Oxidation of 1 with 3‐chloroperbenzoic acid gave 1‐oxide 5 as the major compound along with a trace of 1,2‐dioxide 6.

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