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Syntheses of deuterium labelled atropine and scopolamine

✍ Scribed by Frédéric Balssa; Yves Bonnaire

Publisher
John Wiley and Sons
Year
2009
Tongue
French
Weight
132 KB
Volume
52
Category
Article
ISSN
0022-2135

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✦ Synopsis

Abstract

Easy preparative scale syntheses of deuterium labelled atropine and scopolamine are described. [^2^H~3~]‐atropine and [^2^H~3~]‐scopolamine are obtained in good yield and good isotopic purity in two steps starting from the unlabelled alkaloids. Copyright © 2009 John Wiley & Sons, Ltd.

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