✦ LIBER ✦

Syntheses of [2-14C] 2,5′-anhydro-3′-azido-3′-deoxythymidine and [2-14C] 2,5′-anhydro-3′-azido-2′,3′-dideoxy-5-iodouridine: Inhibitors of human immunodeficiency virus (HIV-1)

✍ Scribed by Tai-Shun Lin; Mao-Chin Liu; E. Michael August; Evelyn M. Birks; William H. Prusoff

Publisher: John Wiley and Sons
Year: 1991
Tongue: French
Weight: 300 KB
Volume: 29
Category: Article
ISSN: 0022-2135
DOI: 10.1002/jlcr.2580291208

No coin nor oath required. For personal study only.

✦ Synopsis

Abstract

The syntheses of [2‐^14^C] 2,5′‐anhydro‐3′‐azido‐3′‐deoxythymidine and [2‐^14^C] 2,5′‐anhydro‐3′‐azido‐2′,3′‐dideoxy‐5‐iodouridine in a one pot operation under mild conditions are described.

📜 SIMILAR VOLUMES

Synthesis of [2-14C] 3′-deoxythymidin-2′

Synthesis of [2-14C] 3′-deoxythymidin-2′ -ENE (d4T) and [5–125I] 3′ -azido-2′, 3′-dideoxy-5-iodouridine: Potent inhibitors of human immunodeficiency virus (HIV-1)

✍ Tai-Shun Lin; You-Song Gao; E. Michael August; He-Ying Qian; William H. Prusoff 📂 Article 📅 1989 🏛 John Wiley and Sons 🌐 French ⚖ 235 KB

Synthesis of 2,5-dideoxy-2-C-methyl-d-ar

Synthesis of 2,5-dideoxy-2-C-methyl-d-arabinose derivatives from methyl 2,3-anhydro-5-deoxy-α-d-ribofuranoside

✍ Hiroshi Yamamoto; Hiroshi Sasaki; Saburo Inokawa 📂 Article 📅 1984 🏛 Elsevier Science 🌐 English ⚖ 553 KB

Synthesis of 5′-amino- and 5′-azido-2′,5

Synthesis of 5′-amino- and 5′-azido-2′,5′-dideoxy nucleosides from thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione

✍ A. A. El-Barbary; N. R. El-Brollosy; E. B. Pedersen; C. Nielsen 📂 Article 📅 1995 🏛 Springer Vienna 🌐 English ⚖ 467 KB

Methyl 5-O-tert-butyldiphenylsilyl-2-deo

Methyl 5-O-tert-butyldiphenylsilyl-2-deoxy-D-threo-pentofuranoside; an approach to the syntesis of 3′-substituted-2′,3′-dideoxynucleosides including 3′-azido-3′-deoxythymidine and of 3′-substituted-2′,3′-dideoxy-C-nucleosides

✍ George W.J Fleet; Jong Chan Son 📂 Article 📅 1987 🏛 Elsevier Science 🌐 French ⚖ 322 KB

Synthesis of [2,3,4,5-14C]-1-vinyl-2-pyr

Synthesis of [2,3,4,5-14C]-1-vinyl-2-pyrrolidinone

✍ George A. Digenis; J. S. McClanahan; Pei-Lin Chen 📂 Article 📅 1993 🏛 John Wiley and Sons 🌐 French ⚖ 257 KB 👁 1 views

## Abstract An efficient small scale synthesis of ^14^C labeled 1‐vinyl‐2‐pyrrolidinone (NVP) is described. The cyclization of commercially available [1,2,3,4‐^14^C]‐γ‐aminobutyric acid (GABA) gives [2,3,4,5‐^14^C]‐2‐pyrrolidinone which is vinylized with vinyl acetate via a sodium tetrachloropallad

Synthesis of 2-amino-7-isopropyl-5-OXO-5

Synthesis of 2-amino-7-isopropyl-5-OXO-5H- [1] benzopyrano-[2,3-b] [2-14C]pyridine-3-carboxylic acid (AA-673-14C)

✍ Nobuyoshi Hayashi; Masayuki Imanishi 📂 Article 📅 1986 🏛 John Wiley and Sons 🌐 French ⚖ 119 KB

17-85. Jusohonmachi 2-chome, Yodogawa-ku. Osaka 532, Japan. ## 2-Amino -7-isopropyl-5-0~0-5H-[ 11 benzopyrano[ 2,3-b] pyridine-3-carboxylic acid (AA-673) was found in these laboratories during the course of the studies on antiallergic agents. passive cutaneous anaphylaxis reaction in rats and the