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Structure−Activity Relationship of 3-Substituted N -(Pyridinylacetyl)-4- (8-chloro-5,6-dihydro-11 H -benzo[5,6]cyclohepta[1,2- b ]pyridin-11-ylidene)- piperidine Inhibitors of Farnesyl-Protein Transferase: Design and Synthesis of in Vivo Active Antitumor Compounds

✍ Scribed by Njoroge, F. George; Vibulbhan, Bancha; Rane, Dinananth F.; Bishop, W. Robert; Petrin, Joanne; Patton, Robert; Bryant, Mathew S.; Chen, K.-J.; Nomeir, Amin A.; Lin, C.-C.; Liu, Ming; King, Ivan; Chen, Jianping; Lee, Suining; Yaremko, Bohdan; Dell, Janet; Lipari, Philip; Malkowski, Michael; Li, Zujun; Catino, Joseph; Doll, Ronald J.; Girijavallabhan, V.; Ganguly, Ashit K.

Book ID: 127043849
Publisher: American Chemical Society
Year: 1997
Tongue: English
Weight: 411 KB
Volume: 40
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm970464g

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