✦ LIBER ✦

Structure Based Development of Phenylimidazole-Derived Inhibitors of Indoleamine 2,3-Dioxygenase

✍ Scribed by Kumar, Sanjeev; Jaller, Daniel; Patel, Bhumika; LaLonde, Judith M.; DuHadaway, James B.; Malachowski, William P.; Prendergast, George C.; Muller, Alexander J.

Book ID: 119992465
Publisher: American Chemical Society
Year: 2008
Tongue: English
Weight: 282 KB
Volume: 51
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm800512z

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Structure−Activity Study of Brassinin De

Structure−Activity Study of Brassinin Derivatives as Indoleamine 2,3-Dioxygenase Inhibitors

✍ Gaspari, Paul; Banerjee, Tinku; Malachowski, William P.; Muller, Alexander J.; P 📂 Article 📅 2006 🏛 American Chemical Society 🌐 English ⚖ 183 KB

Gene structure of human indoleamine 2,3-

Gene structure of human indoleamine 2,3-dioxygenase

✍ Akihiko Kadoya; Shigenobu Tone; Hiroyasu Maeda; Yohsuke Minatogawa; Ryo Kido 📂 Article 📅 1992 🏛 Elsevier Science 🌐 English ⚖ 743 KB

Identification of selective inhibitors o

Identification of selective inhibitors of indoleamine 2,3-dioxygenase 2

✍ Bakmiwewa, Supun M.; Fatokun, Amos A.; Tran, Anh; Payne, Richard J.; Hunt, Nicho 📂 Article 📅 2012 🏛 Elsevier Science 🌐 English ⚖ 698 KB

S-Benzylisothiourea derivatives as small

S-Benzylisothiourea derivatives as small-molecule inhibitors of indoleamine-2,3-dioxygenase

✍ Kenji Matsuno; Kazushige Takai; Yoshinobu Isaka; Yuka Unno; Masayuki Sato; Osamu 📂 Article 📅 2010 🏛 Elsevier Science 🌐 English ⚖ 416 KB

S-Benzylisothiourea 3a was discovered by its ability to inhibit indoleamine-2,3-dioxygenase (IDO) in our screening program. Subsequent optimization of the initial hit 3a lead to the identification of sub-lM inhibitors 3r and 10h, both of which suppressed kynurenine production in A431 cells. Synthesi

Novel candesartan derivatives as indolea

Novel candesartan derivatives as indoleamine 2,3-dioxygenase inhibitors

✍ Matsuno, Kenji; Yamazaki, Hiroshi; Isaka, Yoshinobu; Takai, Kazushige; Unno, Yuk 📂 Article 📅 2012 🏛 The Royal Society of Chemistry 🌐 English ⚖ 491 KB

Discovery and structure–activity relatio

Discovery and structure–activity relationships of phenyl benzenesulfonylhydrazides as novel indoleamine 2,3-dioxygenase inhibitors

✍ Cheng, Ming-Fu; Hung, Ming-Shiu; Song, Jen-Shin; Lin, Shu-Yu; Liao, Fang-Yu; Wu, 📂 Article 📅 2014 🏛 Elsevier Science 🌐 English ⚖ 398 KB