✦ LIBER ✦

Structure−Activity Study of Brassinin Derivatives as Indoleamine 2,3-Dioxygenase Inhibitors

✍ Scribed by Gaspari, Paul; Banerjee, Tinku; Malachowski, William P.; Muller, Alexander J.; Prendergast, George C.; DuHadaway, James; Bennett, Shauna; Donovan, Ashley M.

Book ID: 118237462
Publisher: American Chemical Society
Year: 2006
Tongue: English
Weight: 183 KB
Volume: 49
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm0508888

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

S-Benzylisothiourea derivatives as small

S-Benzylisothiourea derivatives as small-molecule inhibitors of indoleamine-2,3-dioxygenase

✍ Kenji Matsuno; Kazushige Takai; Yoshinobu Isaka; Yuka Unno; Masayuki Sato; Osamu 📂 Article 📅 2010 🏛 Elsevier Science 🌐 English ⚖ 416 KB

S-Benzylisothiourea 3a was discovered by its ability to inhibit indoleamine-2,3-dioxygenase (IDO) in our screening program. Subsequent optimization of the initial hit 3a lead to the identification of sub-lM inhibitors 3r and 10h, both of which suppressed kynurenine production in A431 cells. Synthesi

Synthesis and biological evaluation of n

Synthesis and biological evaluation of novel tryptoline derivatives as indoleamine 2,3-dioxygenase (IDO) inhibitors

✍ Tanaka, Minoru; Li, Xin; Hikawa, Hidemasa; Suzuki, Takafumi; Tsutsumi, Katsuhiko 📂 Article 📅 2013 🏛 Elsevier Science 🌐 English ⚖ 733 KB

Estimation of indoleamine 2,3-dioxygenas

Estimation of indoleamine 2,3-dioxygenase activity as kynurenine to tryptophan ratio in Turkish adolescents

✍ Gözde Girgin; Terken Baydar; Dietmar Fuchs; Orhan Derman; Gönül Şahin 📂 Article 📅 2009 🏛 Elsevier Science 🌐 English ⚖ 85 KB

ChemInform Abstract: Synthesis and Inhib

ChemInform Abstract: Synthesis and Inhibition Study of Monoamine Oxidase, Indoleamine 2, 3-Dioxygenase and Tryptophan 2,3-Dioxygenase by 3,8-Substituted 5H-Indeno[1,2-c]pyridazin-5-one Derivatives.

✍ J. Reniers; C. Meinguet; L. Moineaux; B. Masereel; S. P. Vincent; R. Frederick; 📂 Article 📅 2012 🏛 John Wiley and Sons ⚖ 32 KB

SAR Studies of 3-Cyclopropanecarbonyloxy

SAR Studies of 3-Cyclopropanecarbonyloxy-2-cyclohexen-1-one as Inhibitors of 4-Hydroxyphenylpyruvate Dioxygenase

✍ Yung-Lung Lin; Chung-Shieh Wu; Shean-Woei Lin; Jian-Lin Huang; Yang-Sheng Sun; D 📂 Article 📅 2002 🏛 Elsevier Science 🌐 English ⚖ 151 KB

The first step of the dioxygenation reac

The first step of the dioxygenation reaction carried out by tryptophan dioxygenase and indoleamine 2,3-dioxygenase as revealed by quantum mechanical/molecular mechanical studies

✍ Capece, Luciana (author);Lewis-Ballester, Ariel (author);Batabyal, Dipanwita (au 📂 Article 📅 2010 🏛 John Wiley and Sons 🌐 English ⚖ 588 KB