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Solid-phase synthesis of diverse tetrahydro-1,4-benzodiazepine-2-ones

โœ Scribed by Gurdip Bhalay; Paul Blaney; Vanessa H. Palmer; Anthony D. Baxter


Book ID
108385335
Publisher
Elsevier Science
Year
1997
Tongue
French
Weight
179 KB
Volume
38
Category
Article
ISSN
0040-4039

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## Abstract An efficient solidโ€phase synthetic method for 2,3,4,5โ€Tetrahydroโ€1,4โ€benzodiazepinโ€2,5โ€diones, having amine derivatives on the benzene ring, was developed. This method has been successfully applied to the synthesis of several spatially separated drugโ€like and informationโ€rich smallโ€mole