A solid-phase synthesis ofpolysubstituted 1,5-benzodiazepin-2-ones is described. Resinbound 4-fluoro-3-nitrobanzoic acid was reacted with different ~amino acids, followed by nitro group reduction and formation of the seven-membered ring. Subsequent alkylations at N(5) and N(1) afforded the title com
โฆ LIBER โฆ
Solution-Phase Parallel Synthesis of Diverse 1,5-Benzodiazepin-2-ones
โ Scribed by Zhao, Hai-Yan; Liu, Gang
- Book ID
- 111954688
- Publisher
- American Chemical Society
- Year
- 2007
- Tongue
- English
- Weight
- 333 KB
- Volume
- 9
- Category
- Article
- ISSN
- 1520-4766
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