๐”– Bobbio Scriptorium
โœฆ   LIBER   โœฆ

Solid-Phase Synthesis of 2-Aminoimidazolones

โœ Scribed by Fu, Mengmeng; Fernandez, Monica; Smith, Marie L.; Flygare, John A.


Book ID
118046664
Publisher
American Chemical Society
Year
1999
Tongue
English
Weight
117 KB
Volume
1
Category
Article
ISSN
1523-7060

No coin nor oath required. For personal study only.


๐Ÿ“œ SIMILAR VOLUMES


Rapid assembly of 2-aminoimidazolones on
โœ Kexin Yang; Boliang Lou; Hossain Saneii ๐Ÿ“‚ Article ๐Ÿ“… 2002 ๐Ÿ› Elsevier Science ๐ŸŒ French โš– 173 KB

A straightforward solid-phase synthesis of 2-aminoimidazolone derivatives is described. The synthesis starts with immobilization of thioureas onto solid support, followed by HBTU/DIEA assisted coupling of Boc-protected amino acids. Upon removal of the Boc group, intramolecular cyclization and simult

Solid-phase synthesis of 2-aminoimidazol
โœ David H Drewry; Chiara Ghiron ๐Ÿ“‚ Article ๐Ÿ“… 2000 ๐Ÿ› Elsevier Science ๐ŸŒ French โš– 187 KB

The synthesis of 2-aminoimidazolinones from resin-bound amino acids is described. Reaction of resinbound amino acids with isothiocyanates followed by treatment of the thioureas with Mukaiyama's reagent aorded the corresponding carbodiimides, which reacted with amines to give 2-aminoimidazolinones in

Solid-Phase Synthesis of 2-Aminothiazole
โœ Kearney, Patrick C.; Fernandez, Monica; Flygare, John A. ๐Ÿ“‚ Article ๐Ÿ“… 1998 ๐Ÿ› American Chemical Society ๐ŸŒ English โš– 116 KB
Solid-phase synthesis of ฮ”2-isoxazolines
โœ Jie-Fei Cheng; Adnan M.M. Mjalli ๐Ÿ“‚ Article ๐Ÿ“… 1998 ๐Ÿ› Elsevier Science ๐ŸŒ French โš– 186 KB

Solid-phase synthesis of A2-isoxazolines through a 1,3-dipolar cycioaddition of nitrile oxides is described. The aldoxime is oxidized with commercially available bleach to give the corresponding nitrile oxide, which reacts in situ with dipolarophiles to afford A2-isoxazolines in good yields.