✦ LIBER ✦

Selective agonist binding of (S)-2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid (AMPA) and 2S-(2α,3β,4β)-2-carboxy-4-(1-methylethenyl)-3-pyrrolidineacetic acid (kainate) receptors: a molecular modeling study

✍ Scribed by Olli T Pentikäinen; Luca Settimo; Kari Keinänen; Mark S Johnson

Book ID: 113486910
Publisher: Elsevier Science
Year: 2003
Tongue: English
Weight: 723 KB
Volume: 66
Category: Article
ISSN: 0006-2952
DOI: 10.1016/j.bcp.2003.08.013

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Ab Initio studies of receptor interactio

Ab Initio studies of receptor interactions with AMPA ((S)-2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl) propionic acid ) and Kainic acid (2S-(2α,3β,4β))-2-carboxy-4-(1-methylethenyl)-3-pyrrolidineacetic acid

✍ Elise Champeil; Gloria Proni; Danielle Sapse 📂 Article 📅 2009 🏛 Springer-Verlag 🌐 English ⚖ 685 KB

Synthesis and pharmacology of (RS)-2-ami

Synthesis and pharmacology of (RS)-2-amino-3-(3-hydroxy-5-trifluoromethyl-4-isoxazolyl)propionic acid, a potent AMPA receptor agonist

✍ U Madsen; B Ebert; P Krogsgaard-Larsen; EHF Wong 📂 Article 📅 1992 🏛 Elsevier Science 🌐 French ⚖ 562 KB

Molecular pharmacology of the AMPA agoni

Molecular pharmacology of the AMPA agonist, (S)-2-amino-3-(3-hydroxy-5-phenyl-4-isoxazolyl)propionic acid [(S)-APPA] and the AMPA antagonist, (R)-APPA

✍ Ebert, Bjarke; Madsen, Ulf; Lund, Trine M.; Lenz, Sibylle M.; Krogsgaard-Larsen, 📂 Article 📅 1994 🏛 Elsevier Science 🌐 English ⚖ 682 KB

Studies on an ( S )-2-Amino-3-(3-hydroxy

Studies on an ( S )-2-Amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic Acid (AMPA) Receptor Antagonist IKM-159: Asymmetric Synthesis, Neuroactivity, and Structural Characterization

✍ Juknaitė, Lina; Sugamata, Yutaro; Tokiwa, Kazuya; Ishikawa, Yuichi; Takamizawa, 📂 Article 📅 2013 🏛 American Chemical Society 🌐 English ⚖ 573 KB

AMPA receptor agonists: Resolution, conf

AMPA receptor agonists: Resolution, configurational assignment, and pharmacology of (+)-(S)- and (-)-(R)-2-amino-3-[3-hydroxy-5-(2-pyridyl)-isoxazol-4-yl]-propionic acid (2-Py-AMPA)

✍ Tommy N. Johansen; Bjarke Ebert; Erik Falch; Povl Krogsgaard-Larsen 📂 Article 📅 1997 🏛 John Wiley and Sons 🌐 English ⚖ 173 KB 👁 2 views

We have previously shown that whereas (RS)-2-amino-3-(3-hydroxy-5-phenylisoxazol-4-yl)propionic acid (APPA) shows the characteristics of a partial agonist at (RS)-2-amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic acid (AMPA) receptors, (S)-APPA is a full AMPA receptor agonist and (R)-APPA a weak

Synthesis of deuterium and tritium label

Synthesis of deuterium and tritium labelled (RS)-2-amino-3-(5-tert-butyl-3-hydroxy-4-isoxazolyl)-propionic acid (ATPA), a selective kainic acid receptor agonist

✍ Tommy N. Johansen; Calvin R. Hawes; Gareth J. Ellis; Bjarke Ebert; Tine B. Stens 📂 Article 📅 1999 🏛 John Wiley and Sons 🌐 French ⚖ 315 KB 👁 2 views