In an attempt to discover a high-throughput method for the synthesis of 2,6,9-trisubstituted purines, it was found that microwave irradiation was beneficial in accelerating the nucleophilic displacement of halogens by amines at the C-2 position of the purine nucleus. A method for microwave-assisted
Novel solid-phase preparation of 2,6,9-trisubstituted purines for combinatorial library generation
β Scribed by Peter H Dorff; Ravi S Garigipati
- Publisher
- Elsevier Science
- Year
- 2001
- Tongue
- French
- Weight
- 126 KB
- Volume
- 42
- Category
- Article
- ISSN
- 0040-4039
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