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Novel solid-phase synthesis of 2,6-disubstituted 4(3H)-quinazolinones for combinatorial library generation

✍ Scribed by Csaba Wéber; Attila Bielik; Györgyi I Szendrei; István Greiner

Publisher
Elsevier Science
Year
2002
Tongue
French
Weight
98 KB
Volume
43
Category
Article
ISSN
0040-4039

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✦ Synopsis

A novel procedure for the synthesis of 6-alkoxy-2-amino-4(3H)-quinazolinones from 2,4-dichloro-6-hydroxyquinazoline, amines and alcohols using Wang resin is described.

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