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High specific activity tritium labeling of anti-tumor agent CEP-2563

✍ Scribed by Judith A. Egan; Crist N. Filer; Robert L. Hudkins

Publisher: John Wiley and Sons
Year: 2005
Tongue: French
Weight: 94 KB
Volume: 48
Category: Article
ISSN: 0022-2135
DOI: 10.1002/jlcr.1010

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✦ Synopsis

Ester Methylene-3 H] CEP-2563 (9) was synthesized by the tritiation of precursor 6 with NaB 3 H 4 followed by esterification with BOC-Lys(BOC)-b-Ala-OH and deprotection.

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