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Glycosylated peptoids as prototypical HIV-1 protease inhibitors

✍ Scribed by Uttam K. Saha; René Roy

Publisher: Elsevier Science
Year: 1997
Tongue: French
Weight: 263 KB
Volume: 38
Category: Article
ISSN: 0040-4039
DOI: 10.1016/s0040-4039(97)10028-4

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✦ Synopsis

Using a blockwise approach, N-substituted oligoglycine (NSGs) peptoids bearing Nac.etylglucosamine residues in different position of the side chain were efficiently synthesized by a reiterative strategy involving mono N-alkylation and bromoacetylation.

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