Using a blockwise approach, N-substituted oligoglycine (NSGs) peptoids bearing Nac.etylglucosamine residues in different position of the side chain were efficiently synthesized by a reiterative strategy involving mono N-alkylation and bromoacetylation.
β¦ LIBER β¦
Cycloalkylpiperazines as HIV-1 protease inhibitors: enhanced oral absorption
β Scribed by B. Moon Kim; Ben E. Evans; Kevin F. Gilbert; Colleen M. Hanifin; Joseph P. Vacca; Stuart R. Michelson; Paul L. Darke; Joan A. Zugay; Emilio A. Emini; William Schleif; Jiunn H. Lin; I.-W. Chen; Kari Vastag; Paul S. Anderson; Joel R. Huff
- Publisher
- Elsevier Science
- Year
- 1995
- Tongue
- English
- Weight
- 287 KB
- Volume
- 5
- Category
- Article
- ISSN
- 0960-894X
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