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First synthesis of pyrrolo[1,2:1′,2′]azepino[5,6-b]indole derivatives

✍ Scribed by Julien Perron; Benoı̂t Joseph; Jean-Yves Mérour

Publisher: Elsevier Science
Year: 2003
Tongue: French
Weight: 118 KB
Volume: 44
Category: Article
ISSN: 0040-4039
DOI: 10.1016/s0040-4039(03)01703-9

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✦ Synopsis

A new family of pyrrolo[1,2:1%,2%]azepino [5,6-b]indole derivatives 8,15 related to anthramycin skeleton was prepared in good yield from indole-2-carboxylic acid and b-aminoesters 4 through intramolecular cyclisation.

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