𝔖 Bobbio Scriptorium
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Facile synthesis of [11C]buprenorphine for positron emission tomographic studies of opioid receptors

✍ Scribed by John R. Lever; Samuel M. Mazza; Robert F. Dannals; Hayden T. Ravert; Alan A. Wilson; Henry N. Wagner Jr


Book ID
103922323
Publisher
Elsevier Science
Year
1990
Weight
760 KB
Volume
41
Category
Article
ISSN
0883-2889

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Synthesis of N1β€²-([11C]methyl)naltrindol
✍ John R. Lever; Chris M. Kinter; Hayden T. Ravert; John L. Musachio; William B. M πŸ“‚ Article πŸ“… 1995 πŸ› John Wiley and Sons 🌐 French βš– 508 KB

## Abstract A delta opioid receptor antagonist, N1′‐methylnaltrindole (MeNTI), has been labeled with carbon‐11. The precursor for radiolabeling was prepared in 71% yield by benzylation of the phenolic moiety of naltrindole. Alkylation of the indole nitrogen using [^11^C]iodomethane and aqueous tetr