## N1-(111C]-Methyl>2-Br-LSD ([llC] -MBL) has been developed as a positron emission tomography (PET) imaging agent for serotonin 5-HT2 receptors. In vitro receptor binding assays with nonradioactive MBL show high-affinity binding to serotonin 5-HT2 receptors (Ki = 0.5 nM), a secondary interaction
Synthesis and in vivo characterization of d-(+)-(N1-[11C]methyl)-2-Br-LSD: a radioligand for positron emission tomographic studies of serotonin 5-HT2 receptors
β Scribed by Lever, John R.; Dannals, Robert F.; Wilson, Alan A.; Ravert, Hayden T.; Scheffel, Ursula; Hoffman, Beth J.; Hartig, Paul R.; Wong, Dean F.; Wagner, Henry N.
- Book ID
- 122473437
- Publisher
- Elsevier Science
- Year
- 1989
- Weight
- 890 KB
- Volume
- 16
- Category
- Article
- ISSN
- 0883-2897
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