Preparation of a demonstration library of a,a-disubstituted-a-acylaminoketones, of interest as ecdysone agonists, is described. The five-step synthetic sequence employed a,a-disubstituted amino acids, Grignard reagents and carboxylic acids as building blocks in a strategic combination of solid phase
✦ LIBER ✦
Corrigendum to “Combined solid phase and solution synthesis of a library of α,α-disubstituted-α-acylaminoketones”: [Tetrahedron Lett. 43 (2002) 7495–7498]
✍ Scribed by Javier Garcia; Ernesto Nicolàs; Fernando Albericio; Enrique L. Michelotti; Colin M. Tice
- Publisher
- Elsevier Science
- Year
- 2002
- Tongue
- French
- Weight
- 65 KB
- Volume
- 43
- Category
- Article
- ISSN
- 0040-4039
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